SCHEMBL4032880

SCHEMBL4032880

CCc1nn(C2CC2)cc1C=O

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
DRD2 P14416 1/20 0.30
DRD4 P21917 1/20 0.30
DRD3 P35462 1/20 0.30
AADAT Q8N5Z0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29339717 0.73 RAB9A (0.37) ALDH1A1LMNANPC1MAPTRAB9A
SCHEMBL24014929 0.73 SMN1; SMN2 (0.43) ALDH1A1LMNANPC1MAPTRAB9A
SCHEMBL17196353 0.72 KDR (0.33)
SCHEMBL22979883 0.72 NOTUM (0.38) ALDH1A1LMNANPC1MAPTRAB9A
SCHEMBL25784307 0.72 ELANE (0.39) ALDH1A1LMNANPC1MAPTRAB9A
SCHEMBL25237034 0.71 LRRK2 (0.34) DRD2DRD4DRD3
SCHEMBL22979405 0.69 KDM4E (0.36) ALDH1A1LMNANPC1MAPT
SCHEMBL22979644 0.68 TSHR (0.40) ALDH1A1LMNAMAPT
SCHEMBL29340101 0.68 NPC1 (0.31) ALDH1A1LMNANPC1MAPTRAB9A
SCHEMBL1359607 0.68 LRRK2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725544-B1 3-[4-HETEROCYCLYL-1,2,3-TRIAZOL-1-YL]-N-ARYL-BENZAMIDES AS INHIBITORS OF THE CYTOKINES PRODUCTION FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES BOEHRINGER INGELHEIM PHARMA (US) 2009-05-27 EP disclosed