SCHEMBL4033236

SCHEMBL4033236

Cc1cc(CNc2nccc(Nc3cc(CCc4cccc(F)c4)n[nH]3)n2)no1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 15/20 0.57
FGFR1 P11362 12/20 0.57
KDR P35968 11/20 0.57
INSR P06213 2/20 0.42
PLK4 O00444 1/20 0.38
PAK4 O96013 1/20 0.38
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
SLC2A1 P11166 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4026982 0.90 IGF1R (0.55) IGF1RFGFR1KDRINSR
SCHEMBL3950749 0.88 IGF1R (0.67) IGF1RFGFR1KDRINSRLMNA
SCHEMBL4032312 0.86 IGF1R (0.52) IGF1RFGFR1KDRINSRPLK4
SCHEMBL4031157 0.83 IGF1R (0.78) IGF1RFGFR1KDRINSR
SCHEMBL4032661 0.82 IGF1R (0.59) IGF1RFGFR1KDRINSRPLK4
SCHEMBL5096885 0.77 IGF1R (0.62) IGF1RFGFR1KDRINSR
SCHEMBL5096988 0.76 IGF1R (0.59) IGF1RFGFR1KDRINSR
SCHEMBL3940507 0.76 IGF1R (0.66) IGF1RFGFR1KDRINSR
SCHEMBL4010199 0.75 IGF1R (0.49) IGF1RFGFR1KDRINSR
SCHEMBL4032918 0.75 IGF1R (0.54) IGF1RFGFR1KDRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009019518-A1 PYRIMIDINE COMPOUNDS HAVING A FGFR INHIBITORY EFFECT ASTRAZENECA AB (SE) 2009-02-12 WO disclosed