SCHEMBL4033309

SCHEMBL4033309

Cc1cnc(CNC(C)Cc2ccccn2)c(C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.44
CYP1A2 P05177 3/20 0.40
MAPT P10636 2/20 0.40
CYP2C19 P33261 2/20 0.40
NPC1 O15118 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
RAB9A P51151 1/20 0.40
HTR5A P47898 1/20 0.40
KMT2A Q03164 4/20 0.39
PDE10A Q9Y233 1/20 0.38
MEN1 O00255 2/20 0.37
PIP4K2C Q8TBX8 1/20 0.37
POLB P06746 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032120 0.88 RAB9A (0.39) CYP1A2MAPTCYP2C19NPC1CYP3A4
SCHEMBL23023058 0.75 SIGMAR1 (0.64) CYP1A2MAPTPOLBCYP2D6TSHR
SCHEMBL2085719 0.73 CXCR4 (0.48) CXCR4CYP1A2MAPTCYP2C19NPC1
SCHEMBL4033313 0.72 CXCR4 (0.49) CXCR4CYP1A2CYP2C19CYP3A4KMT2A
SCHEMBL19214862 0.70 CYP1A2 (0.59) CYP1A2CYP2C19NPC1RAB9AALDH1A1
SCHEMBL13188544 0.69 TAAR1 (0.52) CYP1A2MAPTCYP2C19POLBCYP2D6
SCHEMBL2086487 0.68 CXCR4 (0.38) CXCR4PIP4K2CACHEALDH1A1
SCHEMBL2083874 0.68 CXCR4 (0.38) CXCR4CYP1A2MAPTCYP2C19NPC1
Hydrochloric Acid SCHEMBL11524829 0.68 TAAR1 (0.53) CYP1A2MAPTCYP2C19POLBCYP2D6
SCHEMBL19214816 0.68 HRH1 (0.51) CYP1A2MAPTCYP2C19POLBCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed