SCHEMBL4033313

SCHEMBL4033313

Cc1cnc(CNCC(C)c2ccccn2)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 4/20 0.49
PTGFR P43088 1/20 0.35
KMT2A Q03164 2/20 0.35
DUSP3 P51452 1/20 0.35
PTPN11 Q06124 1/20 0.35
SCN8A Q9UQD0 1/20 0.34
LMNA P02545 1/20 0.34
P2RX3 P56373 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
TSHR P16473 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032125 0.88 CXCR4 (0.38) CXCR4PTGFRKMT2ASCN8ATSHR
Ammonia Solution, Strong SCHEMBL5574435 0.75 CXCR4 (0.50) CXCR4KMT2ADUSP3PTPN11SCN8A
SCHEMBL2086487 0.74 CXCR4 (0.38) CXCR4ALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL4033309 0.72 CXCR4 (0.44) CXCR4KMT2AALDH1A1CYP1A2CYP2C19
SCHEMBL2087023 0.72 CXCR4 (0.52) CXCR4KMT2ADUSP3PTPN11SCN8A
SCHEMBL2084301 0.70 CXCR4 (0.55) CXCR4KMT2ADUSP3PTPN11SCN8A
SCHEMBL5574432 0.70 CXCR4 (0.48) CXCR4KMT2ADUSP3PTPN11SCN8A
SCHEMBL11175372 0.69 TAAR1 (0.50) PTGFRLMNAALDH1A1CYP1A2CYP2C19
SCHEMBL31256717 0.69 CXCR4 (0.40) CXCR4ALDH1A1CYP1A2
SCHEMBL2083874 0.68 CXCR4 (0.38) CXCR4KMT2ACYP1A2CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed