SCHEMBL4033607

SCHEMBL4033607

NC(=O)CC1(c2ccccc2)CCN(C(=O)CCc2ccccc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
FKBP1A P62942 1/20 0.53
POLB P06746 2/20 0.51
TSHR P16473 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NAAA Q02083 1/20 0.49
ME2 P23368 1/20 0.48
ME1 P48163 1/20 0.48
ME3 Q16798 1/20 0.48
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
GFER P55789 1/20 0.47
MAPT P10636 1/20 0.47
ALDH1A1 P00352 1/20 0.46
OPRD1 P41143 1/20 0.46
OPRK1 P41145 1/20 0.46
EPHX2 P34913 1/20 0.46
KDM1A O60341 1/20 0.46
SIGMAR1 Q99720 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12195386 0.81 NPC1 (0.56) NPC1TDP1FKBP1APOLBTSHR
SCHEMBL7381627 0.80 NPC1 (0.65) NPC1TDP1FKBP1APOLBTSHR
SCHEMBL2472654 0.79 TSHR (0.48) NPC1TDP1FKBP1APOLBTSHR
SCHEMBL3934544 0.79 NPFFR1 (0.60) POLBTSHRKMT2AMEN1MAPT
SCHEMBL2700497 0.79 NPC1 (0.63) NPC1TDP1FKBP1APOLBTSHR
SCHEMBL7131839 0.77 NPC1 (0.86) NPC1TDP1FKBP1APOLBTSHR
SCHEMBL21077873 0.76 MAOA (0.41) TSHRL3MBTL1KMT2AMEN1EPHX2
SCHEMBL16565921 0.76 P2RX7 (0.53) KMT2AMAPTALDH1A1OPRD1OPRK1
SCHEMBL23718995 0.76 NPC1 (0.60) NPC1TDP1FKBP1APOLBTSHR
SCHEMBL13593925 0.76 NPC1 (0.60) NPC1TDP1FKBP1APOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501467-A4 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION BRISTOL MYERS SQUIBB CO (US) 2009-08-19 EP disclosed
EP-1501467-A2 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION Bristol-Myers Squibb Company (US) 2005-02-02 EP disclosed
WO-2003088908-A2 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION BRISTOL-MYERS SQUIBB COMPANY (US) 2003-10-30 WO disclosed