SCHEMBL4034054

SCHEMBL4034054

Cc1cc(Cl)cnc1CN(Cc1ncccc1CC(C)c1ccccc1)C1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GPR119 Q8TDV5 9/20 0.39
CACNB4 O00305 1/20 0.38
CACNA1A O00555 1/20 0.38
CACNA1G O43497 1/20 0.38
CACNG3 O60359 1/20 0.38
CACNA1F O60840 1/20 0.38
CACNA1H O95180 1/20 0.38
CACNB3 P54284 1/20 0.38
CACNA2D1 P54289 1/20 0.38
CACNG7 P62955 1/20 0.38
CACNA1B Q00975 1/20 0.38
CACNA1D Q01668 1/20 0.38
CACNB1 Q02641 1/20 0.38
CACNG1 Q06432 1/20 0.38
CACNB2 Q08289 1/20 0.38
CACNA1S Q13698 1/20 0.38
CACNA1C Q13936 1/20 0.38
CACNA1E Q15878 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035722 0.94 MEN1 (0.39) MEN1KMT2AGPR119CACNB4CACNA1A
SCHEMBL2085708 0.86 MEN1 (0.40) MEN1KMT2AGPR119FNTAFNTB
SCHEMBL2084970 0.84 MEN1 (0.44) MEN1KMT2AGPR119CACNB4CACNA1A
SCHEMBL4032061 0.81 SLC6A2 (0.41)
SCHEMBL2084600 0.81 MEN1 (0.42) MEN1KMT2AGPR119CACNB4CACNA1A
SCHEMBL4034887 0.79 NR1D1 (0.40) MEN1KMT2AGPR119FNTAFNTB
SCHEMBL2084094 0.79 MEN1 (0.42) MEN1KMT2AGPR119FNTAFNTB
SCHEMBL2082179 0.78 GPR119 (0.51) MEN1KMT2AGPR119POLB
SCHEMBL2084109 0.78 MEN1 (0.41) MEN1KMT2AGPR119
SCHEMBL2086372 0.77 MEN1 (0.45) MEN1KMT2AGPR119POLBUSP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed