SCHEMBL4035722

SCHEMBL4035722

Cc1cc(Cl)cnc1CN(Cc1ncccc1CC(C)c1ccc(F)cc1)C1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GPR119 Q8TDV5 5/20 0.37
TP53 P04637 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP3A5 P20815 1/20 0.37
FNTA P49354 2/20 0.36
FNTB P49356 2/20 0.36
CACNB4 O00305 1/20 0.35
CACNA1A O00555 1/20 0.35
CACNA1G O43497 1/20 0.35
CACNG3 O60359 1/20 0.35
CACNA1F O60840 1/20 0.35
CACNA1H O95180 1/20 0.35
CACNB3 P54284 1/20 0.35
CACNA2D1 P54289 1/20 0.35
CACNG7 P62955 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1D Q01668 1/20 0.35
CACNB1 Q02641 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4034054 0.94 MEN1 (0.40) MEN1KMT2AGPR119TP53CYP3A4
SCHEMBL2084094 0.84 MEN1 (0.42) MEN1KMT2AGPR119TP53FNTA
SCHEMBL2085708 0.84 MEN1 (0.40) MEN1KMT2AGPR119TP53CYP3A4
SCHEMBL2084970 0.79 MEN1 (0.44) MEN1KMT2AGPR119TP53FNTA
SCHEMBL2084600 0.78 MEN1 (0.42) MEN1KMT2AGPR119TP53CACNB4
SCHEMBL4034887 0.78 NR1D1 (0.40) MEN1KMT2AGPR119TP53CYP3A4
SCHEMBL2083669 0.77 MEN1 (0.44) MEN1KMT2AGPR119TP53SQOR
SCHEMBL2082179 0.77 GPR119 (0.51) MEN1KMT2AGPR119POLB
SCHEMBL2084109 0.76 MEN1 (0.41) MEN1KMT2AGPR119LMNA
SCHEMBL5054917 0.75 SMO (0.35) MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed