SCHEMBL4034569

SCHEMBL4034569

Cc1cc(Nc2nc(NCc3cccnc3)ncc2Cl)n[nH]1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 9/20 0.66
FGFR1 P11362 8/20 0.66
KDR P35968 7/20 0.66
INSR P06213 1/20 0.66
BCL6 P41182 1/20 0.57
NTRK1 P04629 3/20 0.53
PAK4 O96013 7/20 0.52
PLK4 O00444 6/20 0.52
AURKA O14965 4/20 0.52
AURKB Q96GD4 3/20 0.52
JAK2 O60674 2/20 0.52
RET P07949 2/20 0.52
FLT3 P36888 2/20 0.52
JAK3 P52333 2/20 0.52
PTK2 Q05397 2/20 0.52
TNK2 Q07912 2/20 0.52
DAPK3 O43293 1/20 0.52
ABL1 P00519 1/20 0.52
LCK P06239 1/20 0.52
FYN P06241 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4031791 0.88 IGF1R (0.79) IGF1RFGFR1KDRINSRBCL6
SCHEMBL2123750 0.87 IGF1R (0.85) IGF1RFGFR1KDRINSRNTRK1
SCHEMBL4038016 0.87 IGF1R (0.79) IGF1RFGFR1KDRINSRBCL6
SCHEMBL2122674 0.87 IGF1R (0.58) IGF1RFGFR1KDRINSRBCL6
SCHEMBL4036060 0.83 IGF1R (0.55) IGF1RFGFR1KDRINSRNTRK1
SCHEMBL4037067 0.82 IGF1R (0.69) IGF1RFGFR1KDRINSR
SCHEMBL4035128 0.82 IGF1R (0.61) IGF1RFGFR1KDRINSRPAK4
SCHEMBL3338201 0.81 NTRK1 (0.59) IGF1RFGFR1KDRINSRNTRK1
SCHEMBL3335945 0.81 NTRK1 (0.72) IGF1RFGFR1KDRINSRNTRK1
SCHEMBL12430659 0.80 NTRK1 (0.74) IGF1RFGFR1KDRINSRNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1456182-B1 PYRIMIDINE DERIVATIVES AS MODULATORS OF INSULINE-LIKE GROWTH FACTOR-1 RECEPTOR (IGF-I) ASTRAZENECA AB (SE) 2009-03-11 EP disclosed