SCHEMBL4034771

SCHEMBL4034771

CC(C)(C)c1ccc(S(=O)(=O)N2CCN(S(=O)(=O)c3ccc4ncccc4c3)C(C(=O)NC3CC3)C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
EPHX2 P34913 1/20 0.47
CHRM5 P08912 3/20 0.46
LMNA P02545 1/20 0.46
GLA P06280 1/20 0.46
PKM P14618 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TSHR P16473 1/20 0.43
GFER P55789 1/20 0.43
MMP1 P03956 1/20 0.43
MMP3 P08254 1/20 0.43
MMP7 P09237 1/20 0.43
MMP9 P14780 1/20 0.43
MMP13 P45452 1/20 0.43
CHRM1 P11229 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CCR4 P51679 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041721 0.87 GAA (0.51) ALDH1A1CHRM5LMNAGLAPKM
SCHEMBL4041974 0.87 GAA (0.51) ALDH1A1CHRM5LMNAGLAPKM
SCHEMBL4034808 0.87 GAA (0.51) ALDH1A1CHRM5LMNAGLAPKM
SCHEMBL4034764 0.86 TSHR (0.61) ALDH1A1EPHX2LMNAHTTSMN1; SMN2
SCHEMBL4035266 0.86 ALDH1A1 (0.47) ALDH1A1CHRM5LMNAGLAPKM
SCHEMBL4033038 0.86 ALDH1A1 (0.47) ALDH1A1CHRM5LMNAGLAPKM
SCHEMBL4040978 0.86 ALDH1A1 (0.47) ALDH1A1CHRM5LMNAGLAPKM
SCHEMBL4037945 0.86 ALDH1A1 (0.47) ALDH1A1CHRM5LMNAGLAPKM
SCHEMBL4035166 0.85 ALDH1A1 (0.51) ALDH1A1CHRM5LMNAGLAPKM
SCHEMBL4036566 0.83 ALDH1A1 (0.62) ALDH1A1LMNAGLAPKMHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed