SCHEMBL4035166

SCHEMBL4035166

CC(C)(C)c1ccc(S(=O)(=O)N2CCN(S(=O)(=O)c3ccc4ncccc4c3)C(C(=O)NCc3ccncc3)C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
HTT P42858 3/20 0.51
LMNA P02545 1/20 0.51
GLA P06280 1/20 0.51
PKM P14618 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CHRM1 P11229 1/20 0.46
GAA P10253 1/20 0.45
USP2 O75604 1/20 0.44
HSD11B1 P28845 2/20 0.44
KMT2A Q03164 1/20 0.44
NPC1 O15118 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CHRM5 P08912 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041721 0.88 GAA (0.51) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4034808 0.88 GAA (0.51) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4041974 0.88 GAA (0.51) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4036566 0.87 ALDH1A1 (0.62) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4037945 0.87 ALDH1A1 (0.47) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4032653 0.87 MAPK1 (0.51) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4040978 0.87 ALDH1A1 (0.47) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4035266 0.87 ALDH1A1 (0.47) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4033038 0.87 ALDH1A1 (0.47) ALDH1A1HTTLMNAGLAPKM
SCHEMBL4034771 0.85 ALDH1A1 (0.53) ALDH1A1HTTLMNAGLAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed