SCHEMBL4035556

SCHEMBL4035556

Cc1cccnc1CNCCc1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.55
ALDH1A1 P00352 2/20 0.55
CYP2C19 P33261 1/20 0.55
HRH3 Q9Y5N1 1/20 0.54
CYP2D6 P10635 2/20 0.54
LMNA P02545 2/20 0.53
ALOX15 P16050 2/20 0.53
TAAR1 Q96RJ0 1/20 0.53
SCN8A Q9UQD0 1/20 0.51
CHRM2 P08172 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
KDM4E B2RXH2 1/20 0.45
DPP7 Q9UHL4 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30481998 0.86 SCN8A (0.55) CYP1A2ALDH1A1CYP2C19SCN8ACHRM2
SCHEMBL1392847 0.80 CHRM2 (0.70) CYP1A2ALDH1A1CYP2C19HRH3CYP2D6
SCHEMBL2082460 0.80 NOS3 (0.45) SCN8AKDM4ENPC1RAB9A
SCHEMBL1921574 0.78 HRH3 (0.70) CYP1A2ALDH1A1CYP2C19HRH3CYP2D6
SCHEMBL4620705 0.78 SCN8A (0.42) ALDH1A1SCN8ACHRM2
SCHEMBL2854302 0.77 CYP1A2 (0.56) CYP1A2ALDH1A1CYP2C19HRH3CYP2D6
SCHEMBL23428554 0.76 SCN8A (0.44) HRH3SCN8ACHRM2NPC1
2-Pyridinecarboxaldehyde SCHEMBL25378590 0.76 SCN8A (0.46) CYP1A2CYP2C19SCN8ACHRM2KDM4E
SCHEMBL23053146 0.76 CYP1A2 (0.69) CYP1A2ALDH1A1CYP2C19HRH3CYP2D6
SCHEMBL17591665 0.76 ALOX15 (0.46) CYP1A2ALDH1A1CYP2C19HRH3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed