SCHEMBL4042715

SCHEMBL4042715

CSCCC1NC2(CCN(SC(=O)O)CC2)N(Cc2ccccc2C#N)C1=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
TSHR P16473 3/20 0.33
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GALR3 O60755 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
BRD4 O60885 1/20 0.33
DPP4 P27487 2/20 0.32
CHRM1 P11229 1/20 0.32
P2RX7 Q99572 1/20 0.32
MAPT P10636 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
CHRM4 P08173 1/20 0.31
FAP Q12884 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3916351 0.90 GAA (0.34) FEN1GAAKMT2ATSHRLMNA
SCHEMBL4032369 0.89 GAA (0.32) FEN1GAAKMT2ATSHRLMNA
SCHEMBL4036440 0.87 TSHR (0.34) GAAKMT2ATSHRLMNASMN1; SMN2
SCHEMBL4035595 0.87 CCR5 (0.38) FEN1TSHROPRM1OPRL1DPP4
SCHEMBL3925602 0.87 GAA (0.36) GAAKMT2ATSHRLMNASMN1; SMN2
SCHEMBL4037470 0.85 GAA (0.44) GAAKMT2ATSHRLMNAALDH1A1
SCHEMBL4035028 0.85 FAAH (0.38) GAATSHRSMN1; SMN2ALDH1A1MAPT
SCHEMBL4038594 0.84 P2RX7 (0.33) GAAKMT2ATSHRLMNASMN1; SMN2
SCHEMBL4040064 0.83 CHRM3 (0.39) FEN1GAAKMT2AOPRM1OPRL1
Benzamide SCHEMBL4033416 0.82 DPP4 (0.33) GAAKMT2ATSHRLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed