SCHEMBL4039787

SCHEMBL4039787

Nc1cc(C2CCN(Cc3ccccc3)C2)c2nc(N)c3cncn3c2n1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.39
HTR6 P50406 5/20 0.38
DRD2 P14416 3/20 0.38
DRD4 P21917 3/20 0.38
DRD3 P35462 3/20 0.38
PDE8B O95263 2/20 0.38
ROCK2 O75116 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
USP30 Q70CQ3 2/20 0.36
ACHE P22303 2/20 0.35
BCHE P06276 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CCR2 P41597 1/20 0.35
ROCK1 Q13464 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039782 0.83 HTR6 (0.39) MCHR1HTR6DRD2DRD4DRD3
SCHEMBL6696801 0.72 ROCK2 (0.48) ROCK2ACHEBCHEHRH3CCR2
Ammonia Solution, Strong SCHEMBL28610050 0.67 ROCK2 (0.47) HTR6ROCK2MEN1KMT2AUSP30
SCHEMBL4896796 0.66 MEN1 (0.54) HTR6DRD2DRD4DRD3MEN1
SCHEMBL4896785 0.66 MEN1 (0.54) HTR6DRD2DRD4DRD3MEN1
SCHEMBL73760 0.65 HRH3 (0.53) DRD2DRD4DRD3MEN1KMT2A
SCHEMBL14724848 0.64 OPRM1 (0.53) HTR6DRD2DRD4DRD3MEN1
SCHEMBL1546751 0.63 HTR6 (0.50) HTR6DRD2DRD4MEN1KMT2A
SCHEMBL7969987 0.62 LCK (0.66) ROCK2KMT2AACHEBCHECCR2
SCHEMBL1546893 0.62 USP30 (0.48) HTR6DRD2DRD4DRD3USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1066286-B1 HETEROCYCLO-SUBSTITUTED IMIDAZOPYRAZINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2009-04-29 EP claimed