SCHEMBL404075

SCHEMBL404075

COC(=O)c1ccc(-c2nc(C)ccc2C(=O)OCc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.52
KDM4E B2RXH2 3/20 0.48
KMT2A Q03164 3/20 0.48
HPGD P15428 3/20 0.48
GAA P10253 3/20 0.48
MEN1 O00255 1/20 0.48
MAPT P10636 6/20 0.48
RAB9A P51151 4/20 0.48
ALDH1A1 P00352 5/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
HTT P42858 2/20 0.47
NPC1 O15118 2/20 0.47
LMNA P02545 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A3 Q01959 1/20 0.47
TSHR P16473 3/20 0.46
MAPK1 P28482 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
DHODH Q02127 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL402418 0.81 TDP1 (0.46) KDM4EKMT2AHPGDGAAMEN1
SCHEMBL22388846 0.78 KMT2A (0.76) PKMKDM4EKMT2AHPGDGAA
SCHEMBL17158280 0.77 TDP1 (0.53) PKMKDM4EKMT2AHPGDGAA
SCHEMBL20201203 0.77 ALDH1A1 (0.55) KMT2AHPGDMEN1MAPTRAB9A
SCHEMBL6647268 0.75 RAB9A (0.53) KMT2AHPGDGAAMAPTRAB9A
SCHEMBL401600 0.75 POLB (0.62) KMT2ARAB9AALDH1A1SMN1; SMN2LMNA
SCHEMBL31414565 0.75 TSHR (0.53) PKMKDM4EKMT2AMAPTRAB9A
Dimethyl Phthalate SCHEMBL7826081 0.74 KMT2A (0.69) PKMKDM4EKMT2AHPGDGAA
SCHEMBL6647657 0.72 PKM (0.61) PKMKDM4EKMT2AHPGDGAA
SCHEMBL6644878 0.72 TSHR (0.48) PKMKDM4EKMT2AHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
CN-101056628-B Ester derivatives and medicinal use thereof JAPAN TOBACCO INC 2011-05-25 CN disclosed
CN-101056628-A Ester derivatives and medicinal use thereof JAPAN TOBACCO INC (JP) 2007-10-17 CN disclosed
EP-1803452-A1 ESTER DERIVATIVE AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2007-07-04 EP disclosed
EP-1803452-A1 ESTER DERIVATIVE AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2007-07-04 EP disclosed
US-20060089392-A1 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2006-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060089392-A1 Ester derivatives and medicinal use thereof MTTP, CETP, LIPA PKM 1414/4885KDM4E 2908/4885KMT2A 3181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.