SCHEMBL4041520

SCHEMBL4041520

CSCCC1NC2(CCN(SOC(=O)Nc3cccc(C)c3)CC2)N(C)C1=O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
GRM5 P41594 1/20 0.35
KMT2A Q03164 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
DCUN1D1 Q96GG9 1/20 0.35
DRD2 P14416 4/20 0.35
DRD4 P21917 4/20 0.35
DRD3 P35462 3/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
CCKBR P32239 1/20 0.34
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3917060 0.83 ALDH1A1 (0.47) ALDH1A1KMT2AL3MBTL1MEN1LMNA
SCHEMBL4032651 0.77 SMN1; SMN2 (0.37) ALDH1A1KMT2AMEN1LMNA
SCHEMBL4036406 0.75 UBE2M (0.39) ALDH1A1BCHEACHEGRM5KMT2A
SCHEMBL4036539 0.74 FAAH (0.38) ALDH1A1KMT2ADCUN1D1DRD2DRD4
SCHEMBL4034635 0.72 HDAC8 (0.35) ALDH1A1KMT2A
SCHEMBL3915996 0.69 HDAC8 (0.36) ALDH1A1KMT2AMEN1
SCHEMBL4035369 0.69 GAA (0.42) ALDH1A1KMT2AL3MBTL1LMNA
SCHEMBL4033021 0.69 HDAC8 (0.34) ALDH1A1KMT2A
SCHEMBL1800547 0.68 TDP1 (0.47) ALDH1A1ACHEKMT2AL3MBTL1MEN1
SCHEMBL4041320 0.68 PLA2G10 (0.38) ALDH1A1KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed
EP-1730144-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5|DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2006-12-13 EP claimed
WO-2005095398-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4.5]DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2005-10-13 WO claimed
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP disclosed
EP-1730144-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5|DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2006-12-13 EP disclosed
WO-2005095398-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4.5]DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2005-10-13 WO disclosed