SCHEMBL4042121

SCHEMBL4042121

CSCCC1NC2(CCN(SC(=O)O)CC2)N(Cc2ccc(F)cc2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
CCR5 P51681 5/20 0.32
CXCR3 P49682 1/20 0.32
HTT P42858 1/20 0.32
GHSR Q92847 1/20 0.32
SIGMAR1 Q99720 2/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
CHRM2 P08172 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CHRM3 P20309 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4037470 0.91 GAA (0.44) GAAKMT2ACCR5CXCR3HTT
SCHEMBL3927067 0.89 GAA (0.37) GAAKMT2ACCR5CXCR3HTT
SCHEMBL4034816 0.88 GAA (0.34) GAAKMT2ACCR5CXCR3HTT
SCHEMBL4035046 0.86 GAA (0.35) GAAKMT2ACCR5CXCR3SIGMAR1
SCHEMBL3919512 0.86 GAA (0.39) GAAKMT2ACCR5CXCR3ALDH1A1
SCHEMBL4033395 0.85 MCHR1 (0.36) GAAKMT2ASIGMAR1CYP3A4CYP2D6
SCHEMBL4040751 0.83 HTT (0.38) HTTPOLB
SCHEMBL4035720 0.83 TP53 (0.35) KMT2ACCR5HTTALDH1A1POLB
SCHEMBL2940213 0.83 RIPK1 (0.42) GAAKMT2AHTTCHRM2CYP3A4
SCHEMBL1801114 0.83 RIPK1 (0.42) GAAKMT2AHTTCHRM2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed