SCHEMBL4037470

SCHEMBL4037470

CSCCC1NC2(CCN(SC(=O)O)CC2)N(Cc2ccccc2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.44
KMT2A Q03164 1/20 0.44
CCR5 P51681 7/20 0.38
CACNA1G O43497 1/20 0.37
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CXCR3 P49682 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042121 0.91 GAA (0.36) GAAKMT2ACCR5ALDH1A1HTT
SCHEMBL4033395 0.90 MCHR1 (0.36) GAAKMT2AACHE
SCHEMBL3918968 0.88 GAA (0.46) GAAKMT2ACCR5CACNA1GMAPT
SCHEMBL4040064 0.88 CHRM3 (0.39) GAAKMT2A
SCHEMBL4035369 0.87 GAA (0.42) GAAKMT2ACCR5CACNA1GMAPT
SCHEMBL4034900 0.86 CXCR3 (0.40) GAACCR5KDM4EALDH1A1LMNA
SCHEMBL4042715 0.85 FEN1 (0.33) GAAKMT2AMAPTTSHRALDH1A1
SCHEMBL4035139 0.85 GAA (0.43) GAAKMT2ACCR5CACNA1GMAPT
SCHEMBL3925963 0.85 GAA (0.47) GAAKMT2ACCR5CACNA1GMAPT
SCHEMBL2935516 0.83 KMT2A (0.49) GAAKMT2ACCR5CACNA1GMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed