SCHEMBL4033395

SCHEMBL4033395

CSCCC1NC2(CCN(SC(=O)O)CC2)N(Cc2ccc3ccccc3c2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.36
SIGMAR1 Q99720 2/20 0.36
KMT2A Q03164 4/20 0.36
GAA P10253 1/20 0.36
ACHE P22303 1/20 0.35
MEN1 O00255 3/20 0.35
MMP13 P45452 1/20 0.34
GRM2 Q14416 1/20 0.34
CCR3 P51677 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CAPN1 P07384 1/20 0.33
FAAH O00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4037470 0.90 GAA (0.44) KMT2AGAAACHE
SCHEMBL3994486 0.89 MCHR1 (0.37) MCHR1SIGMAR1KMT2AGAAACHE
SCHEMBL4206788 0.89 KMT2A (0.35) MCHR1SIGMAR1KMT2AGAAACHE
SCHEMBL1810683 0.88 ACHE (0.36) MCHR1SIGMAR1KMT2AGAAACHE
SCHEMBL4046162 0.87 MCHR1 (0.38) MCHR1SIGMAR1KMT2AGAAACHE
SCHEMBL3995879 0.87 KMT2A (0.38) MCHR1SIGMAR1KMT2AGAAACHE
SCHEMBL4042121 0.85 GAA (0.36) SIGMAR1KMT2AGAACYP3A4CYP2D6
SCHEMBL1809029 0.85 TSHR (0.43) MCHR1KMT2AGAAMEN1
SCHEMBL4040064 0.84 CHRM3 (0.39) SIGMAR1KMT2AGAACCR3FAAH
Dimethylamine SCHEMBL3987722 0.83 ACHE (0.35) MCHR1SIGMAR1KMT2AGAAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed