SCHEMBL4043020

SCHEMBL4043020

CN(C)CCNc1cc(NN)ncn1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DNM2 P50570 7/20 0.65
HRH4 Q9H3N8 1/20 0.63
HRH3 Q9Y5N1 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAP4K4 O95819 1/20 0.47
GAA P10253 1/20 0.41
ALPG P10696 1/20 0.41
EGFR P00533 2/20 0.40
AURKA O14965 1/20 0.40
KIT P10721 1/20 0.40
FLT3 P36888 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
CHEK1 O14757 1/20 0.38
LCK P06239 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12497656 0.81 DNM2 (0.62) DNM2HRH4HRH3CYP2C19MAP4K4
SCHEMBL17581278 0.79 DNM2 (0.60) DNM2HRH4HRH3CYP2C19MAP4K4
SCHEMBL1774003 0.78 HRH4 (1.00) DNM2HRH4HRH3CYP2C19MAP4K4
SCHEMBL17300725 0.77 DNM2 (0.57) DNM2HRH4HRH3CYP2C19MAP4K4
SCHEMBL12410840 0.77 DNM2 (0.57) DNM2HRH4HRH3CYP2C19MAP4K4
SCHEMBL13472373 0.74 DNM2 (0.55) DNM2HRH4HRH3CYP2C19MAP4K4
SCHEMBL4076540 0.74 L3MBTL1 (0.42) GAAEGFRCHEK1
SCHEMBL27523685 0.72 EGFR (0.51) DNM2HRH4CYP2C19MAP4K4EGFR
SCHEMBL2948693 0.72 HRH4 (0.55) DNM2HRH4HRH3CYP2C19MAP4K4
SCHEMBL15834613 0.71 DNM2 (0.59) DNM2HRH4EGFRLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed