SCHEMBL4043256

SCHEMBL4043256

CC(C)CC(NC(=O)Oc1ccc2ccccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1ccccn1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSK P43235 16/20 0.41
CTSL P07711 13/20 0.39
CTSS P25774 9/20 0.39
CTSB P07858 4/20 0.39
CTSV O60911 2/20 0.36
MC4R P32245 1/20 0.35
MC3R P41968 1/20 0.35
MC1R Q01726 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CASP1 P29466 1/20 0.34
CASP3 P42574 1/20 0.34
CASP7 P55210 1/20 0.34
CASP6 P55212 1/20 0.34
CASP8 Q14790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043226 0.95 CTSK (0.40) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4047535 0.92 MC4R (0.38) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4045521 0.91 CTSK (0.43) CTSKCTSLCTSSCTSBKDM4E
SCHEMBL4050724 0.90 CTSK (0.39) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4048011 0.89 CTSK (0.40) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4044864 0.89 CTSK (0.43) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4050151 0.89 CTSK (0.41) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4047693 0.88 CTSK (0.40) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4041738 0.88 CTSK (0.43) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4046943 0.88 CTSK (0.50) CTSKCTSLCTSSCTSBMC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed