SCHEMBL4046943

SCHEMBL4046943

CC(C)CC(NC(=O)Oc1ccc2ccccc2c1)C(=O)N1CCC2C1C(=O)CN2C(=O)c1ccccn1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 14/20 0.50
CTSS P25774 6/20 0.42
CTSL P07711 6/20 0.42
CTSB P07858 3/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
CASP1 P29466 2/20 0.36
CASP3 P42574 2/20 0.36
CASP7 P55210 2/20 0.36
CASP6 P55212 2/20 0.36
CASP8 Q14790 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MC4R P32245 1/20 0.35
MC3R P41968 1/20 0.35
MC1R Q01726 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050228 0.94 CTSK (0.49) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4043597 0.92 CTSK (0.41) CTSKCTSSCTSLGAASMN1; SMN2
SCHEMBL4045333 0.91 CTSK (0.53) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4043401 0.89 CTSK (0.47) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4046025 0.88 CTSK (0.49) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4041452 0.88 CTSK (0.49) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4042251 0.88 CTSK (0.50) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4043256 0.88 CTSK (0.41) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4044026 0.87 CTSK (0.49) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4045412 0.87 CTSK (0.48) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed