SCHEMBL4043732

SCHEMBL4043732

CCOC(=O)c1ccc(OCCCN2CCOCC2)c(OC)c1N

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
CYP2D6 P10635 1/20 0.48
TSHR P16473 1/20 0.48
KDM4E B2RXH2 4/20 0.47
TDP1 Q9NUW8 1/20 0.47
POLB P06746 2/20 0.47
GAA P10253 2/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 1/20 0.46
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
THRB P10828 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
HTR1A P08908 1/20 0.44
HTR2A P28223 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044992 0.84 ALDH1A1 (0.54) ALDH1A1CYP2D6TSHRKDM4ETDP1
SCHEMBL31620999 0.83 CYP2D6 (0.50) ALDH1A1CYP2D6TSHRKDM4ETDP1
SCHEMBL11385195 0.81 HTR1A (0.52) ALDH1A1KDM4ESMN1; SMN2HTR1AHTR2A
SCHEMBL6442660 0.80 LMNA (0.51) ALDH1A1CYP2D6TSHRKDM4ETDP1
SCHEMBL3534600 0.80 LMNA (0.51) ALDH1A1CYP2D6TSHRKDM4ETDP1
SCHEMBL7315768 0.79 ALDH1A1 (0.64) ALDH1A1CYP2D6KDM4ETDP1POLB
SCHEMBL3531517 0.78 SMN1; SMN2 (0.63) ALDH1A1CYP2D6TSHRKDM4ETDP1
SCHEMBL4047895 0.78 KDM4E (0.53) ALDH1A1CYP2D6TSHRKDM4ETDP1
SCHEMBL6447779 0.78 SMN1; SMN2 (0.63) ALDH1A1CYP2D6TSHRKDM4ETDP1
SCHEMBL23965931 0.78 CYP2D6 (0.53) ALDH1A1CYP2D6TSHRKDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103719-A1 SUBSTITUTED 4-(INDOL-3-YL)QUINAZOLINES AND USE AND PRODUCTION THEREOF FREIE UNIVERSITÄT BERLIN (DE) 2009-08-27 WO disclosed