SCHEMBL4044959

SCHEMBL4044959

O=C(O)N1CC(c2nc3nccnc3[nH]2)C1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.40
HTR2B P41595 1/20 0.37
PDE10A Q9Y233 12/20 0.36
PBK Q96KB5 4/20 0.35
DGAT2 Q96PD7 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050701 0.76 PBK (0.41) EGLN1PBK
SCHEMBL1299454 0.70 HTR2B (0.52) HTR2B
SCHEMBL4055604 0.69 METAP2 (0.35) PBK
SCHEMBL1304590 0.67 PDE10A (0.43) PDE10A
SCHEMBL1740554 0.67 CYP2C9 (0.46) PDE10A
SCHEMBL30515605 0.67 KDM4E (0.53) EGLN1
SCHEMBL21435110 0.66 HPGDS (0.34) HTR2B
SCHEMBL1740546 0.65 PDE10A (0.40) PDE10A
SCHEMBL21435247 0.65 HPGDS (0.35) HTR2B
SCHEMBL2595525 0.64 HTR2B (0.50) HTR2BPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed