SCHEMBL4055604

SCHEMBL4055604

CC1(C)CC(c2nc3nccnc3[nH]2)C1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.35
METAP1 P53582 1/20 0.35
PBK Q96KB5 4/20 0.32
CDK1 P06493 1/20 0.30
CDK9 P50750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050701 0.80 PBK (0.41) METAP2METAP1PBKCDK1CDK9
SCHEMBL4054581 0.77 ADORA1 (0.40) METAP2METAP1PBK
SCHEMBL4059999 0.77 METAP2 (0.38) METAP2METAP1PBK
SCHEMBL7300780 0.65 METAP2 (0.33) METAP2METAP1
SCHEMBL813686 0.64 METAP2 (0.44) METAP2METAP1CDK1
SCHEMBL4052899 0.60 NPC1 (0.38) CDK1
SCHEMBL976118 0.60 METAP2 (0.48) METAP2METAP1CDK1
SCHEMBL14409054 0.60 METAP2 (0.44) METAP2METAP1
Zarzissine SCHEMBL1514280 0.60 NUDT1 (0.50) METAP2METAP1
SCHEMBL6012369 0.60 METAP2 (0.44) METAP2METAP1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed