SCHEMBL4046834

SCHEMBL4046834

N#Cc1cccc2c1OC=CO2

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.44
ESR2 Q92731 1/20 0.37
TSHR P16473 1/20 0.35
CYP11B1 P15538 5/20 0.34
CYP11B2 P19099 5/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
HTT P42858 1/20 0.32
MCL1 Q07820 1/20 0.31
MTNR1A P48039 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
HIF1A Q16665 1/20 0.30
AR P10275 1/20 0.30
MAP2K1 Q02750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18936028 0.83 TRPA1 (0.44) TRPA1ESR2TSHRCYP11B1CYP11B2
SCHEMBL18936192 0.77 TRPA1 (0.40) TRPA1ESR2TSHRCYP11B1CYP11B2
SCHEMBL9618582 0.76
SCHEMBL17069064 0.73 ABCG2 (0.44) TRPA1TSHRCYP11B1CYP11B2
SCHEMBL7128137 0.73 ITGB2 (0.44) TRPA1CYP11B1CYP11B2HTTMTNR1A
SCHEMBL17289161 0.73 TRPA1 (0.40) TRPA1ESR2TSHRCA1CA2
SCHEMBL24010287 0.71 TRPA1 (0.56) TRPA1ESR2TSHRCA1CA2
SCHEMBL728135 0.70 MTNR1A (0.34) MTNR1A
SCHEMBL15320700 0.67 TRPA1 (0.38) TRPA1HTT
SCHEMBL18112905 0.67 TRPA1 (0.51) TRPA1ESR2TSHRAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010532-A1 TRYCLIC NITROGEN CONTAINING COMPOUNDS AND THEIR USE AS ANTIBACTERIALS Glaxo Group Limited (GB) 2009-01-07 EP claimed
WO-2007122258-A1 TRYCLIC NITROGEN CONTAINING COMPOUNDS AND THEIR USE AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2007-11-01 WO claimed