SCHEMBL4046896

SCHEMBL4046896

CCC(CCc1sc2c(c1C#N)CCC(NCC1CCc3ccccc31)C2)CNC(=O)c1ccccc1O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 2/20 0.37
MAPT P10636 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SAE1 Q9UBE0 1/20 0.36
UBA2 Q9UBT2 1/20 0.36
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TAS1R3 Q7RTX0 2/20 0.33
TAS1R1 Q7RTX1 2/20 0.33
TAS1R2 Q8TE23 2/20 0.33
MEN1 O00255 1/20 0.33
ALOX12 P18054 1/20 0.33
KMT2A Q03164 1/20 0.33
PIN1 Q13526 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HTT P42858 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4037340 0.87 GCGR (0.44) GCGRMAPTNPSR1SAE1UBA2
SCHEMBL4038702 0.84 MAPT (0.38) GCGRMAPTNPSR1SAE1UBA2
SCHEMBL4045769 0.82 TP53 (0.35) GCGRMAPTNPSR1SAE1UBA2
SCHEMBL4043069 0.81 GCGR (0.43) GCGRMAPTNPSR1SAE1UBA2
SCHEMBL4037334 0.80 NPSR1 (0.36) GCGRMAPTNPSR1SAE1UBA2
SCHEMBL4041950 0.80 MAPT (0.36) GCGRMAPTNPSR1SAE1UBA2
SCHEMBL4045782 0.80 MAPT (0.36) GCGRMAPTNPSR1SAE1UBA2
SCHEMBL4355052 0.79 MTNR1B (0.44) GCGRMAPTNPSR1SAE1UBA2
SCHEMBL6315675 0.77 NPC1 (0.35) MAPTNPSR1SAE1UBA2ALDH1A1
SCHEMBL4042444 0.76 ALDH1A1 (0.39) GCGRMAPTNPSR1SAE1UBA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1549655-B1 SUBSTITUTED BICYCLIC THIOPHENE DERIVATIVES, COMPOSTIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO INC (US) 2009-01-21 EP claimed