SCHEMBL4047993

SCHEMBL4047993

CC1Cc2ccc(C(=O)CCl)cc2CN1C(=O)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ESR1 P03372 3/20 0.36
ESR2 Q92731 3/20 0.36
RAB9A P51151 2/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
DDR1 Q08345 1/20 0.33
DDR2 Q16832 1/20 0.33
NPC1 O15118 1/20 0.33
HTT P42858 1/20 0.33
PTPN11 Q06124 1/20 0.33
PDK2 Q15119 2/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4227747 0.79 ESR1 (0.40) ESR1ESR2OPRM1OPRD1OPRK1
SCHEMBL1366031 0.78 ESR1 (0.48) ALDH1A1MAPTSMN1; SMN2ESR1ESR2
SCHEMBL1367390 0.77 ESR1 (0.64) ALDH1A1MAPTSMN1; SMN2ESR1ESR2
SCHEMBL8248218 0.75 PNMT (0.46)
SCHEMBL8241195 0.75 HTR2C (0.44) MAPTSMN1; SMN2RAB9ANPC1PDK2
SCHEMBL1366408 0.74 ESR1 (0.52) ALDH1A1MAPTSMN1; SMN2ESR1ESR2
SCHEMBL4050990 0.73 MCHR1 (0.55) MCHR1
SCHEMBL4565375 0.73 MCHR1 (0.54) MCHR1
SCHEMBL2310619 0.71 ALDH1A1 (0.37) ALDH1A1MAPTSMN1; SMN2RAB9AKDM4E
SCHEMBL5737230 0.70 CA1 (0.42) ALDH1A1MAPTSMN1; SMN2RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103478-A1 PYRIDONE AND PYRIDAZINONE DERIVATIVES AS MCH ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-08-27 WO disclosed