SCHEMBL4048357

SCHEMBL4048357

Cc1ccc(C)c(S(=O)(=O)NCCN2C[C@@H]3C[C@H]2CN3C(=O)[C@@H](NC(=O)c2cc3ccccc3[nH]2)C(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.38
PLD1 Q13393 1/20 0.36
CYP51A1 Q16850 1/20 0.35
STAT6 P42226 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
PLD2 O14939 1/20 0.34
CNR2 P34972 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CCKBR P32239 1/20 0.33
PYGL P06737 1/20 0.33
AKR1C3 P42330 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050835 0.90 DRD2 (0.39) DRD2PLD1CYP51A1STAT6CNR2
SCHEMBL4059459 0.86 PYGL (0.38) DRD2PLD1CYP51A1STAT6PYGL
SCHEMBL4051527 0.86 DRD3 (0.39) DRD2PLD1CYP51A1STAT6PYGL
SCHEMBL4058360 0.84 DRD2 (0.36) DRD2PLD1CYP51A1STAT6ALDH1A1
SCHEMBL4051134 0.83 DRD2 (0.38) DRD2PLD1CYP51A1STAT6CNR2
SCHEMBL19856897 0.82 DRD2 (0.41) DRD2CYP51A1STAT6KDM4ECNR2
SCHEMBL19856899 0.82 DRD2 (0.41) DRD2CYP51A1STAT6KDM4ECNR2
SCHEMBL8004902 0.81 DRD2 (0.38) DRD2CYP51A1STAT6CCKBRPYGL
SCHEMBL1549547 0.80 PDGFRB (0.46) DRD2CYP51A1STAT6PYGLAKR1C3
SCHEMBL1549906 0.80 DRD2 (0.42) DRD2CYP51A1STAT6KDM4ECNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO claimed
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed