SCHEMBL4059459

SCHEMBL4059459

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2CCNS(=O)(=O)c1cc(Cl)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PYGL P06737 4/20 0.38
DRD3 P35462 2/20 0.38
BCAT1 P54687 2/20 0.37
DRD2 P14416 1/20 0.37
CYP51A1 Q16850 5/20 0.37
PLD1 Q13393 1/20 0.36
OPRK1 P41145 1/20 0.36
ALOX15 P16050 1/20 0.35
STAT6 P42226 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051527 0.94 DRD3 (0.39) PYGLDRD3BCAT1DRD2CYP51A1
SCHEMBL4058360 0.92 DRD2 (0.36) PYGLDRD3DRD2CYP51A1PLD1
SCHEMBL4057673 0.90 PYGL (0.39) PYGLDRD3BCAT1DRD2CYP51A1
SCHEMBL4048357 0.86 DRD2 (0.38) PYGLDRD2CYP51A1PLD1STAT6
SCHEMBL7993594 0.86 PYGL (0.40) PYGLBCAT1DRD2CYP51A1
SCHEMBL4057362 0.84 PYGL (0.39) PYGLDRD3BCAT1DRD2CYP51A1
SCHEMBL4051117 0.84 ALOX15 (0.42) PYGLBCAT1CYP51A1ALOX15
SCHEMBL4347129 0.83 PYGL (0.39) PYGLBCAT1DRD2CYP51A1PLD1
SCHEMBL4056168 0.83 ALDH1A1 (0.42) PYGLBCAT1DRD2CYP51A1STAT6
SCHEMBL19856896 0.83 PYGL (0.43) PYGLDRD3DRD2CYP51A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed