SCHEMBL4048581

SCHEMBL4048581

CCCCc1c(N)cccc1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 5/20 0.47
TSHR P16473 5/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HSD17B10 Q99714 1/20 0.42
PDE7A Q13946 1/20 0.41
MAPT P10636 4/20 0.40
CYP3A4 P08684 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GPR35 Q9HC97 1/20 0.39
ALDH1A1 P00352 4/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
RECQL P46063 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4938054 0.95 TDP1 (0.46) TDP1TSHRSMN1; SMN2HSD17B10PDE7A
SCHEMBL7166893 0.90 TDP1 (0.46) TDP1TSHRSMN1; SMN2HSD17B10PDE7A
SCHEMBL27321459 0.83 TSHR (0.55) TDP1TSHRSMN1; SMN2HSD17B10MAPT
SCHEMBL1668133 0.83 TDP1 (0.48) TDP1TSHRSMN1; SMN2HSD17B10PDE7A
SCHEMBL10777337 0.82 TDP1 (0.48) TDP1TSHRSMN1; SMN2HSD17B10MAPT
SCHEMBL27884727 0.81 GPR35 (0.50) TDP1TSHRSMN1; SMN2HSD17B10CYP3A4
SCHEMBL17242666 0.81 TSHR (0.45) TDP1TSHRMAPTCYP3A4CYP1A2
SCHEMBL3393735 0.80 GPR35 (0.46) TDP1TSHRSMN1; SMN2PDE7AMAPT
SCHEMBL7342960 0.79 TSHR (0.48) TDP1TSHRSMN1; SMN2MAPTCYP3A4
Alcohol SCHEMBL11148831 0.79 FBP1 (0.46) TDP1TSHRSMN1; SMN2HSD17B10PDE7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101891680-B Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-29 CN disclosed
CN-103641765-A Modulators of ATP-binding cassette transporters VERTEX PHARMA 2014-03-19 CN disclosed
CN-101935301-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2013-10-16 CN disclosed
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
EP-2032583-A1 NEW CHEMICAL COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2009-03-11 EP disclosed
WO-2007144370-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-12-21 WO disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed
CN-1671700-A Substituted alkylamine derivatives and methods of use AMGEN INC (US) 2005-09-21 CN disclosed
US-4395572-A Process for preparing N-alkyl-nitroanilines UNION CARBIDE CORPORATION (US) 1983-07-26 US disclosed
US-4289907-A Process for preparing N-alkyl-nitroanilines UNION CARBIDE CORPORATION (US) 1981-09-15 US disclosed