SCHEMBL4049678

SCHEMBL4049678

N=C(N)c1cc(C(=O)O)ccc1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.49
WDR5 P61964 1/20 0.47
F10 P00742 2/20 0.47
F11 P03951 2/20 0.47
F7 P08709 2/20 0.47
TTR P02766 1/20 0.46
ALDH1A1 P00352 1/20 0.46
PTPRC P08575 2/20 0.45
CYP2C8 P10632 1/20 0.45
CYP2C9 P11712 1/20 0.45
KDM4E B2RXH2 1/20 0.45
KMO O15229 1/20 0.44
FOLH1 Q04609 1/20 0.44
PLAU P00749 1/20 0.44
PLAT P00750 1/20 0.44
DHODH Q02127 1/20 0.44
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
MAP4K4 O95819 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5215160 0.86 BCAT2 (0.61) BCAT2TTRALDH1A1PTPRCCYP2C8
SCHEMBL594370 0.84 FOLH1 (0.59) TTRALDH1A1PTPRCCYP2C8CYP2C9
Water SCHEMBL28745832 0.82 FOLH1 (0.57) TTRALDH1A1PTPRCCYP2C8CYP2C9
SCHEMBL29562805 0.82 TTR (0.52) TTRALDH1A1PTPRCCYP2C8CYP2C9
SCHEMBL22729968 0.82 TTR (0.52) TTRALDH1A1PTPRCCYP2C8CYP2C9
SCHEMBL27736136 0.79 CYP2C8 (0.71) TTRALDH1A1CYP2C8CYP2C9KDM4E
SCHEMBL3104353 0.79 KDM4C (0.53) TTRALDH1A1PTPRCCYP2C8CYP2C9
SCHEMBL1569116 0.79 EGFR (0.57) TTRALDH1A1CYP2C8CYP2C9KDM4E
SCHEMBL5248866 0.78 KDM4E (0.48) ALDH1A1KDM4EPLAUPRSS1PRSS2
SCHEMBL28791455 0.78 CYP2C8 (0.50) TTRALDH1A1PTPRCCYP2C8CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824825-A4 SUBSTITUTED PYRIDOXINES AS ANTI-PLATELET AGENTS MEDICURE INT INC (BB) 2009-07-08 EP disclosed
EP-1824825-A1 SUBSTITUTED PYRIDOXINES AS ANTI-PLATELET AGENTS Medicure International Inc. (BB) 2007-08-29 EP disclosed
WO-2006045203-A1 SUBSTITUTED PYRIDOXINES AS ANTI-PLATELET AGENTS MEDICURE INTERNATIONAL INC. (CA) 2006-05-04 WO disclosed