SCHEMBL4050226

SCHEMBL4050226

CC(C)Cn1c(=O)[nH]c2cnc(-c3cccc(O)c3)nc21

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.49
MTOR P42345 1/20 0.49
USP1 O94782 16/20 0.47
PIK3CD O00329 1/20 0.44
B3GNT2 Q9NY97 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15206153 0.78 PIK3CA (0.59) ADORA3MTORUSP1PIK3CD
SCHEMBL300868 0.77 PIK3CD (0.71) PIK3CD
SCHEMBL28028896 0.76 PIK3CD (0.49) MTORPIK3CD
SCHEMBL4051247 0.75 PIK3CD (0.43) ADORA3PIK3CD
SCHEMBL15206336 0.74 JAK2 (0.55) ADORA3MTORPIK3CD
SCHEMBL29829189 0.74 JAK2 (0.55) ADORA3MTORPIK3CD
SCHEMBL18865991 0.74 USP1 (0.80) USP1
SCHEMBL29691064 0.74 USP1 (0.80) USP1
SCHEMBL7215331 0.73 ADORA3 (0.68) ADORA3USP1
SCHEMBL4050613 0.72 PIK3CA (0.53) MTORUSP1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078018-A1 HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND USE THEREOF AS PROTEIN KINASE INHIBITORS Signal Pharmaceuticals LLC (US) 2009-07-15 EP disclosed
WO-2008051494-A1 HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND USE THEREOF AS PROTEIN KINASE INHIBITORS SIGNAL PHARMACEUTICALS, LLC (US) 2008-05-02 WO disclosed