SCHEMBL4051074

SCHEMBL4051074

CCOC(=O)/C(=C/I)C(O)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
CYP1A2 P05177 2/20 0.50
LMNA P02545 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ALDH1A1 P00352 3/20 0.41
CES2 O00748 1/20 0.39
ACHE P22303 1/20 0.39
CES1 P23141 1/20 0.39
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
CASP3 P42574 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
SENP7 Q9BQF6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049872 1.00 MAPT (0.50) MAPTMEN1KMT2ACYP1A2LMNA
SCHEMBL4061472 0.88 DHODH (0.44) MAPTMEN1KMT2ACYP1A2LMNA
SCHEMBL4048528 0.88 DHODH (0.44) MAPTMEN1KMT2ACYP1A2LMNA
SCHEMBL4060289 0.85 ALDH1A1 (0.44) MAPTMEN1KMT2ACYP1A2LMNA
SCHEMBL4062017 0.85 MEN1 (0.50) MAPTMEN1KMT2ACYP1A2LMNA
SCHEMBL4057202 0.85 MEN1 (0.50) MAPTMEN1KMT2ACYP1A2LMNA
SCHEMBL4056870 0.85 ALDH1A1 (0.44) MAPTMEN1KMT2ACYP1A2LMNA
SCHEMBL4051755 0.85 MEN1 (0.49) MAPTMEN1KMT2ALMNAGAA
SCHEMBL4061773 0.85 MEN1 (0.49) MAPTMEN1KMT2ALMNAGAA
SCHEMBL4053169 0.85 NPSR1 (0.50) MAPTMEN1KMT2ANPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110655-A1 NOVEL BETA SUBSTITUTED MORITA-BAYLIS-HILLMAN DERIVATIVES SUNGKYUNKWAN UNIVERSITY FOUNDATION FOR CORPORATE COLLABORATION (KR) 2009-09-11 WO claimed
WO-2009110655-A1 NOVEL BETA SUBSTITUTED MORITA-BAYLIS-HILLMAN DERIVATIVES SUNGKYUNKWAN UNIVERSITY FOUNDATION FOR CORPORATE COLLABORATION (KR) 2009-09-11 WO disclosed