SCHEMBL4053169

SCHEMBL4053169

CCOC(=O)/C(=C/I)C(O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.50
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
GPR35 Q9HC97 1/20 0.39
POLB P06746 3/20 0.38
PPARG P37231 3/20 0.38
FFAR1 O14842 2/20 0.38
EPHX2 P34913 1/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 1/20 0.38
HSP90AA1 P07900 1/20 0.38
CRHBP P24387 1/20 0.38
KMT2A Q03164 1/20 0.38
CRHR2 Q13324 1/20 0.38
GAA P10253 1/20 0.37
ALDH1A1 P00352 2/20 0.37
CASP1 P29466 1/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051074 0.85 MAPT (0.50) NPSR1CES2CES1MAPTKDM4E
SCHEMBL4049872 0.85 MAPT (0.50) NPSR1CES2CES1MAPTKDM4E
SCHEMBL4048528 0.84 DHODH (0.44) NPSR1CES2CES1POLBMAPT
SCHEMBL4061472 0.84 DHODH (0.44) NPSR1CES2CES1POLBMAPT
SCHEMBL4062017 0.82 MEN1 (0.50) NPSR1CES2CES1GPR35MAPT
SCHEMBL4060289 0.82 ALDH1A1 (0.44) NPSR1POLBMAPTKDM4EMEN1
SCHEMBL4057202 0.82 MEN1 (0.50) NPSR1CES2CES1GPR35MAPT
SCHEMBL4056870 0.82 ALDH1A1 (0.44) NPSR1POLBMAPTKDM4EMEN1
SCHEMBL15917904 0.82 CASP1 (0.51) NPSR1CES2CES1GPR35POLB
SCHEMBL4061773 0.81 MEN1 (0.49) POLBMAPTMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110655-A1 NOVEL BETA SUBSTITUTED MORITA-BAYLIS-HILLMAN DERIVATIVES SUNGKYUNKWAN UNIVERSITY FOUNDATION FOR CORPORATE COLLABORATION (KR) 2009-09-11 WO claimed
WO-2009110655-A1 NOVEL BETA SUBSTITUTED MORITA-BAYLIS-HILLMAN DERIVATIVES SUNGKYUNKWAN UNIVERSITY FOUNDATION FOR CORPORATE COLLABORATION (KR) 2009-09-11 WO disclosed