SCHEMBL4051885

SCHEMBL4051885

COc1ccc(CC#N)c2c1oc1ccc(C(F)(F)F)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 4/20 0.37
CYP17A1 P05093 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
HSD17B10 Q99714 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
PIM1 P11309 2/20 0.34
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
PIM3 Q86V86 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
CASP1 P29466 1/20 0.33
IDH1 O75874 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
GAK O14976 1/20 0.32
EGFR P00533 1/20 0.32
PDE5A O76074 1/20 0.32
BCL9 O00512 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050927 0.85 CYP17A1 (0.39) CYP17A1CYP19A1CYP11B1CYP11B2HSD17B10
SCHEMBL13693817 0.85 PON1 (0.40) CYP17A1CYP19A1CYP11B1CYP11B2HSD17B10
SCHEMBL4011420 0.79 CYP17A1 (0.47) CYP17A1CYP19A1CYP11B1CYP11B2HSD17B10
SCHEMBL13693816 0.75 GAK (0.38) HSD17B10ALDH1A1HPGDPIM1CSNK2A2
SCHEMBL5022806 0.74 TBK1 (0.47) HSD17B10ALDH1A1HPGDPIM1PIM2
SCHEMBL4062570 0.74 ESRRA (0.37) ESRRAIDH1PDE5AMAPT
SCHEMBL4239976 0.72 PDE4A (0.39) ESRRAHSD17B10ALDH1A1HPGDPIM1
SCHEMBL4051687 0.71 MAOA (0.51) HSD17B10ALDH1A1HPGDRAB9AGAA
SCHEMBL9989279 0.67 SCN9A (0.46) HSD17B10CASP1RAB9AGAAMAPT
SCHEMBL25786471 0.67 DAO (0.43) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed