SCHEMBL4239976

SCHEMBL4239976

COc1ccc(C2(C#N)CCC(=O)CC2)c2c1oc1ccc(C(F)(F)F)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
PIM1 P11309 8/20 0.34
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 1/20 0.33
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
KCNQ4 P56696 1/20 0.33
KCNMA1 Q12791 1/20 0.33
KCNQ5 Q9NR82 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
ESRRA P11474 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053847 0.84 CCR2 (0.33) PDE4APDE4BPDE4CPDE4DPIM1
SCHEMBL4012783 0.83 MAOA (0.43) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL4060397 0.83 DDB1 (0.33) PDE4BPIM1DDB1CRBNHRH4
SCHEMBL4062007 0.81 HRH4 (0.31) HRH4
SCHEMBL4060696 0.80 HRH4 (0.37) HRH4
SCHEMBL4541496 0.77 PIM1 (0.31) PIM1ESRRAMEN1NPC1RAB9A
SCHEMBL4541501 0.77 PIM1 (0.31) PIM1ESRRAMEN1NPC1RAB9A
SCHEMBL4235894 0.77 HRH4 (0.35) HRH4
SCHEMBL4051885 0.72 ESRRA (0.37) PIM1ALDH1A1HPGDHSD17B10ESRRA
SCHEMBL5022806 0.72 TBK1 (0.47) PDE4APDE4BPDE4CPDE4DPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed