SCHEMBL4053445

SCHEMBL4053445

CC(C)(C)N(C(=O)O)c1ccc(C(F)(F)F)cc1CO

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
POLQ O75417 2/20 0.38
KLF10 Q13118 1/20 0.37
APP P05067 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
TACR1 P25103 2/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
USP2 O75604 1/20 0.35
CYP2C19 P33261 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
LSS P48449 1/20 0.35
FFAR4 Q5NUL3 1/20 0.34
CES2 O00748 2/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17507930 0.79 ALDH1A1 (0.51) POLQAPPKDM4EALDH1A1HPGD
SCHEMBL17507931 0.77 KDM4E (0.47) POLQAPPKDM4EALDH1A1HPGD
SCHEMBL1208112 0.75 MEN1 (0.37) CYP3A4ALDH1A1HPGDCYP2C19
SCHEMBL10758967 0.74 PPARA (0.37) APPKDM4EALDH1A1HPGDHSD17B10
SCHEMBL2497436 0.72 EPHX2 (0.44) APPALDH1A1CES2MTOR
SCHEMBL9752985 0.71 PSEN1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL23636332 0.70 TP53 (0.48) KDM4EALDH1A1CES2
SCHEMBL10233691 0.70 ESR1 (0.43) CYP3A4CYP2D6POLQKLF10CYP2C19
SCHEMBL19534969 0.70 HSD11B1 (0.40)
SCHEMBL2116911 0.69 PDCD1 (0.44) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694658-B1 METHOD FOR THE PRODUCTION OF A THIAZOLO [3,4,5-DE] [4,1]BENZOTHIAZEPINE-TYPE PRODUCT AVENTIS PHARMA SA (FR) 2009-02-25 EP claimed