SCHEMBL4054967

SCHEMBL4054967

COC(=O)C1CC(C#N)(c2ccc(OC3CCCC3)c3oc4ccc([N+](=O)[O-])cc4c23)CCC1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 14/20 0.37
PDE4B Q07343 14/20 0.37
PDE4C Q08493 14/20 0.37
PDE4D Q08499 14/20 0.37
CYP19A1 P11511 4/20 0.34
MEN1 O00255 1/20 0.33
PTGES O14684 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
PTGS1 P23219 1/20 0.33
CYP2C19 P33261 1/20 0.33
PTGS2 P35354 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053847 0.77 CCR2 (0.33) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL4051064 0.77 ALDH1A1 (0.34) ALDH1A1CYP3A4MAPTCYP2C19KMT2A
SCHEMBL4012666 0.77 PDE4B (0.37) PDE4APDE4BPDE4CPDE4DCYP19A1
SCHEMBL2868054 0.72 MAPT (0.39) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL5703617 0.72 PDE4A (0.68) PDE4APDE4BPDE4CPDE4D
SCHEMBL4377016 0.71 CYP19A1 (0.41) CYP19A1MEN1PTGESALDH1A1CYP1A2
SCHEMBL4055340 0.69 CYP19A1 (0.43) CYP19A1MEN1PTGESALDH1A1CYP1A2
SCHEMBL6816264 0.69 PDE4A (0.59) PDE4APDE4BPDE4CPDE4D
SCHEMBL4061843 0.69 CYP19A1 (0.41) PDE4APDE4BPDE4CPDE4DCYP19A1
SCHEMBL4033691 0.69 CYP19A1 (0.43) CYP19A1MEN1PTGESALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed