SCHEMBL4051064

SCHEMBL4051064

COC(=O)C1CC(C#N)(c2ccc(OC)c3c2c2cc([N+](=O)[O-])ccc2n3C)CCC1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 4/20 0.34
POLB P06746 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
PKM P14618 1/20 0.33
HTT P42858 1/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
HTR2A P28223 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4059484 0.88 PSEN1 (0.41) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL4050626 0.85 PDE4A (0.39) ALDH1A1SMN1; SMN2MAPTSIGMAR1HTT
SCHEMBL4054967 0.77 PDE4A (0.37) ALDH1A1SMN1; SMN2MAPTNPSR1L3MBTL1
SCHEMBL4241620 0.76 PSEN1 (0.35) MAPTPSEN1PSEN2APH1BNCSTN
SCHEMBL2868054 0.76 MAPT (0.39) ALDH1A1SMN1; SMN2MAPTPSEN1PSEN2
SCHEMBL4050217 0.75 BACE1 (0.32) ALDH1A1SMN1; SMN2MAPTSIGMAR1HTR1A
SCHEMBL521209 0.73 PDE4B (0.42) KMT2A
SCHEMBL6617848 0.72 PDE4A (0.39) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6601490 0.72 PDE4B (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL13693820 0.71 PDE4A (0.41) ALDH1A1SMN1; SMN2HTTHTR2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed