SCHEMBL4054974

SCHEMBL4054974

Cc1nn2c(=O)n(Cc3ccccc3)c(C(NCCNC(=O)OC(C)(C)C)C(C)C)nc2c1Cl

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.39
BRD4 O60885 8/20 0.37
P2RX7 Q99572 1/20 0.36
GNRHR P30968 1/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2A P29274 1/20 0.35
MALT1 Q9UDY8 1/20 0.35
IDO1 P14902 1/20 0.35
P2RX3 P56373 1/20 0.34
BCHE P06276 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4054984 1.00 KIF11 (0.39) KIF11BRD4P2RX7GNRHRADORA3
SCHEMBL4050591 0.95 KIF11 (0.41) KIF11BRD4P2RX7GNRHRADORA3
SCHEMBL4055834 0.95 KIF11 (0.41) KIF11BRD4P2RX7GNRHRADORA3
SCHEMBL4056718 0.95 KIF11 (0.41) KIF11BRD4ADORA3
SCHEMBL4056720 0.95 KIF11 (0.41) KIF11BRD4ADORA3
SCHEMBL4049089 0.87 KIF11 (0.39) KIF11BRD4GNRHRADORA3
SCHEMBL4250470 0.85 GNRHR (0.39) KIF11BRD4GNRHRMALT1IDO1
SCHEMBL4250472 0.85 GNRHR (0.39) KIF11BRD4GNRHRMALT1IDO1
SCHEMBL4048206 0.82 KIF11 (0.51) KIF11
SCHEMBL4048203 0.82 KIF11 (0.51) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074677-A2 PYRAZOLOTRIAZINES 4SC AG (DE) 2009-06-18 WO disclosed
EP-2070932-A1 Pyrazolotriazines 4SC AG (DE) 2009-06-17 EP disclosed