SCHEMBL4055057

SCHEMBL4055057

Oc1cccc2c1[nH]c1ccc(F)cc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.66
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
PLA2G7 Q13093 3/20 0.44
KIF11 P52732 1/20 0.44
ACHE P22303 1/20 0.44
MAPT P10636 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
USP2 O75604 1/20 0.43
METAP2 P50579 1/20 0.42
CHUK O15111 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
MAPK1 P28482 2/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28761777 0.82 AR (0.70) ARGAAACHEMEN1KMT2A
SCHEMBL27919630 0.79 AR (0.66) ARALDH1A1KDM4EGAAPLA2G7
SCHEMBL2324939 0.79 AR (1.00) ARKDM4EMEN1KMT2ACHUK
SCHEMBL25783735 0.79 KIF11 (0.62) ARALDH1A1KDM4EGLAGAA
SCHEMBL26511308 0.79 KDM4E (0.49) ARALDH1A1KDM4EGLAGAA
SCHEMBL6759889 0.78 PBRM1 (0.57) ARALDH1A1KDM4EGLAGAA
SCHEMBL329557 0.77 AR (0.62) ARALDH1A1KDM4EHTTKIF11
SCHEMBL23875434 0.77 AR (0.60) ARALDH1A1KDM4EKIF11ACHE
SCHEMBL23875528 0.77 TUBB4A (0.51) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL17613793 0.77 ACHE (0.47) ALDH1A1KDM4EGLAGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed