SCHEMBL4057043

SCHEMBL4057043

c1cc2c(s1)C(NC1=NCCO1)CC2

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 13/20 0.50
ADRA2B P18089 13/20 0.50
ADRA2C P18825 13/20 0.50
ADRA1A P35348 5/20 0.50
TAAR1 Q96RJ0 7/20 0.36
HTR1A P08908 2/20 0.36
DRD2 P14416 1/20 0.36
HTR7 P34969 1/20 0.36
GMNN O75496 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
OPRK1 P41145 1/20 0.36
HIF1A Q16665 1/20 0.36
NISCH Q9Y2I1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1723548 0.74 ADRA2B (0.84) ADRA2AADRA2BADRA2CADRA1A
SCHEMBL11332296 0.74 ADRA2A (0.62) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL1724062 0.67 ADRA2A (1.00) ADRA2AADRA2BADRA2CADRA1ATSHR
SCHEMBL4054961 0.66 ADRA2A (0.59) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL4564280 0.66 ADRA2A (0.56) ADRA2AADRA2BADRA2CADRA1A
SCHEMBL14449748 0.65 TAAR1 (0.42) TAAR1HTR1ADRD2HTR7
SCHEMBL10159872 0.65 TAAR1 (0.40) TAAR1HTR1ADRD2HTR7
SCHEMBL2216731 0.65 ADRA2A (0.57) ADRA2AADRA2BADRA2CADRA1ATAAR1
SCHEMBL1218576 0.64 ADRA2A (0.67) ADRA2AADRA2BADRA2CADRA1A
SCHEMBL15975257 0.63 ADRA2A (0.55) ADRA2AADRA2BADRA2CADRA1ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2014168-A1 Insecticidal heterocyclic compounds Bayer CropScience AG (DE) 2009-01-14 EP disclosed
EP-2014168-A1 Insecticidal heterocyclic compounds Bayer CropScience AG (DE) 2009-01-14 EP disclosed
WO-2008155031-A1 HETEROCYCLIC COMPOUNDS FOR INSECTICIDES BAYER CROPSCIENCE AG (DE) 2008-12-24 WO disclosed
WO-2008155031-A1 HETEROCYCLIC COMPOUNDS FOR INSECTICIDES BAYER CROPSCIENCE AG (DE) 2008-12-24 WO disclosed