SCHEMBL4057718

SCHEMBL4057718

OC1C2CC3CC1CC(C14CC5CC(CC(O)(C5)C1)C4)(C3)C2

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.41
CYP2C9 P11712 1/20 0.38
ALDH1A1 P00352 2/20 0.33
HSD11B1 P28845 1/20 0.33
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4057608 0.86 PKM (0.52) PKMALDH1A1HSD11B1PRMT5WDR77
SCHEMBL4065340 0.84 CYP2C9 (0.52) CYP2C9
SCHEMBL3844870 0.82 PKM (0.56) PKMALDH1A1HSD11B1PRMT5WDR77
SCHEMBL4064149 0.82 CYP2C9 (0.48) CYP2C9
SCHEMBL4055873 0.76 PKM (0.40) PKMALDH1A1HSD11B1PRMT5WDR77
SCHEMBL3850543 0.76 PKM (0.50) PKMALDH1A1HSD11B1PRMT5WDR77
SCHEMBL1772242 0.75 CYP2C9 (0.46) PKMCYP2C9HSD11B1
SCHEMBL3841419 0.74 PKM (0.48) PKMALDH1A1HSD11B1PRMT5WDR77
Adamantan-2-Ol SCHEMBL8345108 0.73 CYP2C9 (0.65) PKMCYP2C9HSD11B1
SCHEMBL3843113 0.71 PKM (0.40) PKMCYP2C9ALDH1A1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090030248-A1 Ethynylphenylbiadamantane derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2009-01-29 US disclosed
EP-2014636-A1 Ethynylphenylbiadamantane derivatives Daicel Chemical Industries, Ltd. (JP) 2009-01-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090030248-A1 Ethynylphenylbiadamantane derivatives CHRNA5, CHRNE, ADRA1D PKM 4221/4885CYP2C9 271/4885ALDH1A1 1329/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.