SCHEMBL4058078

SCHEMBL4058078

c1ccc(Cc2ccccc2N(Cc2ccccc2)c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.42
NR3C2 P08235 1/20 0.41
TSHR P16473 2/20 0.40
HTR2A P28223 1/20 0.40
CALM1 P0DP23 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
KCNA3 P22001 1/20 0.39
BCL2 P10415 1/20 0.38
BCL2L1 Q07817 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KCNH2 Q12809 1/20 0.36
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
AOC3 Q16853 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3693511 0.79 TRPM8 (0.50) NR3C2TSHRHDAC1HDAC8HDAC6
SCHEMBL30626413 0.79 BCL2 (0.47) PTPN1TSHRHTR2ACALM1BCL2
SCHEMBL5852076 0.79 BCL2 (0.47) PTPN1TSHRHTR2ACALM1BCL2
SCHEMBL1704796 0.79 PTPN1 (0.45) PTPN1NR3C2TSHRHTR2ACALM1
SCHEMBL918512 0.77 NR3C2 (0.56) NR3C2TSHRCALM1HDAC1HDAC8
SCHEMBL10659836 0.76 BCL2 (0.52) PTPN1HTR2ACALM1BCL2BCL2L1
Ammonia Solution, Strong SCHEMBL28750457 0.76 BCL2 (0.44) PTPN1TSHRHTR2ACALM1BCL2
SCHEMBL9446230 0.75 NR3C2 (0.59) NR3C2TSHRHDAC1HDAC8HDAC6
Bromide SCHEMBL4613403 0.75 NR3C2 (0.55) NR3C2TSHRCALM1HDAC1HDAC8
SCHEMBL9116726 0.75 ALDH1A1 (0.45) NR3C2TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141702-B2 Process for the synthesis of α-substituted acroleins COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-11-28 US claimed
US-20050215829-A1 Tandem hydroformylation and Mannich reaction sequence in the presence of syngas and formaldehyde, wherein the two catalysts are segregated into two different phases to prevent deactivation of the catalysts by each other, and yielding a highly selective and active catalyst; e.g. ethylene to methacrolein COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2005-09-29 US claimed
WO-2005063668-A1 PROCESS FOR SYNTHESIS OF ALPHA-SUBSTITUTED ACROLEINS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-07-14 WO claimed
EP-2055763-A1 Lubricating oil composition Shell Internationale Research Maatschappij B.V. (NL) 2009-05-06 EP disclosed
US-7141702-B2 Process for the synthesis of α-substituted acroleins COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-11-28 US disclosed
US-20050215829-A1 Tandem hydroformylation and Mannich reaction sequence in the presence of syngas and formaldehyde, wherein the two catalysts are segregated into two different phases to prevent deactivation of the catalysts by each other, and yielding a highly selective and active catalyst; e.g. ethylene to methacrolein COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2005-09-29 US disclosed
WO-2005063668-A1 PROCESS FOR SYNTHESIS OF ALPHA-SUBSTITUTED ACROLEINS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-07-14 WO disclosed
EP-0326223-B1 Copolymer composition SHELL INT RESEARCH (NL) 1996-05-08 EP disclosed
EP-0458814-A1 FLUOROPOLYMER COMPOSITIONS RAYCHEM CORPORATION (US) 1991-12-04 EP disclosed
US-4992499-A Using phenolic compound and aromatic amine SHELL OIL COMPANY (US) 1991-02-12 US disclosed
WO-1990008805-A1 FLUOROPOLYMER COMPOSITIONS RAYCHEM CORPORATION (US) 1990-08-09 WO disclosed
EP-0326223-A2 Copolymer composition SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1989-08-02 EP disclosed