SCHEMBL4058405

SCHEMBL4058405

O=C(/C=C/C(=O)ON1CCCC1)ON1CCCC1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3751257 1.00 KEAP1 (0.33) KEAP1NFE2L2HCAR2ALDH1A1
SCHEMBL5874735 0.97 ALDH1A1 (0.35) KEAP1NFE2L2HCAR2ALDH1A1
SCHEMBL5875212 0.97 ALDH1A1 (0.35) KEAP1NFE2L2HCAR2ALDH1A1
SCHEMBL1934761 0.95 KEAP1 (0.33) KEAP1NFE2L2HCAR2
SCHEMBL10992799 0.91 HCAR2 (0.43) HCAR2ALDH1A1
SCHEMBL3632775 0.91 HCAR2 (0.43) HCAR2ALDH1A1
SCHEMBL10859674 0.89 HCAR2 (0.41) HCAR2
SCHEMBL10859682 0.89 HCAR2 (0.41) HCAR2
SCHEMBL17695729 0.87 NFE2L2 (0.52) KEAP1NFE2L2HCAR2ALDH1A1
SCHEMBL20240604 0.86 GSTP1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009094457-A2 SUBSTITUTED BENZHYDRYLETHERS AUSPEX PHARMACEUTICALS (US) 2009-07-30 WO disclosed
CN-101426778-A N-substituted-azacyclylamines as histamine-3 antagonists WYETH CORP (US) 2009-05-06 CN disclosed
EP-1994022-A2 N-SUBSTITUTED-AZACYCLYLAMINES AS HISTAMINE-3 ANTAGONISTS Wyeth a Corporation of the State of Delaware (US) 2008-11-26 EP disclosed
WO-2007108936-A2 N-SUBSTITUTED-AZACYCLYLAMINES AS HISTAMINE-3 ANTAGONISTS WYETH (US) 2007-09-27 WO disclosed
US-4698430-A ANTIDEPRESSANT A. H. ROBINS COMPANY, INC. (US) 1987-10-06 US disclosed