SCHEMBL4058816

SCHEMBL4058816

CCOC(=O)/C(=C/I)C(O)c1ccc(C#N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 3/20 0.39
KDM4E B2RXH2 3/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
DNTT P04053 1/20 0.39
GPR35 Q9HC97 1/20 0.39
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
FNTA P49354 2/20 0.37
FNTB P49356 2/20 0.37
ALDH1A1 P00352 3/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
GSK3B P49841 1/20 0.36
POLB P06746 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4054818 1.00 PDCD1 (0.41) PDCD1CD274HTTL3MBTL1KDM4E
SCHEMBL4061472 0.84 DHODH (0.44) HTTGAAMAPTALDH1A1POLB
SCHEMBL4048528 0.84 DHODH (0.44) HTTGAAMAPTALDH1A1POLB
SCHEMBL4057202 0.82 MEN1 (0.50) HTTKDM4EGAAMAPTGPR35
SCHEMBL4056870 0.82 ALDH1A1 (0.44) L3MBTL1KDM4EGAAMAPTALDH1A1
SCHEMBL4049872 0.82 MAPT (0.50) HTTKDM4EGAAMAPTALDH1A1
SCHEMBL4051074 0.82 MAPT (0.50) HTTKDM4EGAAMAPTALDH1A1
SCHEMBL4060289 0.82 ALDH1A1 (0.44) L3MBTL1KDM4EGAAMAPTALDH1A1
SCHEMBL4062017 0.82 MEN1 (0.50) HTTKDM4EGAAMAPTGPR35
SCHEMBL4061773 0.81 MEN1 (0.49) GAAMAPTALDH1A1POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110655-A1 NOVEL BETA SUBSTITUTED MORITA-BAYLIS-HILLMAN DERIVATIVES SUNGKYUNKWAN UNIVERSITY FOUNDATION FOR CORPORATE COLLABORATION (KR) 2009-09-11 WO claimed
WO-2009110655-A1 NOVEL BETA SUBSTITUTED MORITA-BAYLIS-HILLMAN DERIVATIVES SUNGKYUNKWAN UNIVERSITY FOUNDATION FOR CORPORATE COLLABORATION (KR) 2009-09-11 WO disclosed