SCHEMBL4059231

SCHEMBL4059231

CC(=O)Nc1ccc(O)cc1N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.55
MAPT P10636 2/20 0.52
POLB P06746 1/20 0.52
RAB9A P51151 1/20 0.52
CA1 P00915 5/20 0.48
CA2 P00918 5/20 0.48
CA9 Q16790 5/20 0.48
ALDH1A1 P00352 3/20 0.48
MEN1 O00255 1/20 0.48
CA12 O43570 1/20 0.48
BRD4 O60885 1/20 0.48
NR1I2 O75469 1/20 0.48
MB P02144 1/20 0.48
CYP1A1 P04798 1/20 0.48
CA3 P07451 1/20 0.48
CYP3A4 P08684 1/20 0.48
RARG P13631 1/20 0.48
TSHR P16473 1/20 0.48
ALOX5AP P20292 1/20 0.48
CA4 P22748 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11512570 0.85 HDAC1 (0.60) NPC1MAPTPOLBRAB9ACA1
SCHEMBL628743 0.82 NPC1 (0.66) NPC1MAPTPOLBRAB9ACA1
SCHEMBL28990133 0.82 NPC1 (0.63) NPC1MAPTPOLBRAB9ACA1
SCHEMBL30354741 0.82 NPC1 (0.63) NPC1MAPTPOLBRAB9ACA1
SCHEMBL31198179 0.81 HDAC1 (0.60) NPC1MAPTPOLBRAB9ACA1
SCHEMBL2767464 0.81 HDAC1 (0.60) NPC1MAPTPOLBRAB9ACA1
SCHEMBL10371584 0.81 NPC1 (0.55) NPC1MAPTPOLBRAB9ACA1
SCHEMBL10371585 0.81 NPC1 (0.55) NPC1MAPTPOLBRAB9ACA1
SCHEMBL9509772 0.81 NPC1 (0.55) NPC1MAPTPOLBRAB9ACA1
SCHEMBL11027199 0.81 HDAC1 (0.60) NPC1MAPTRAB9ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547713-B2 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2009-06-16 US claimed
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2006-05-25 US claimed
US-7547713-B2 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2009-06-16 US disclosed
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2006-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives PTGS2, PTGES2, PTGES NPC1 4539/4885MAPT 3965/4885POLB 1417/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.