SCHEMBL4059920

SCHEMBL4059920

NCCN(Cc1ccccc1)c1nc(C(=O)NCc2cccc(Cl)c2Cl)c(O)c2ncccc12

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.47
ADORA1 P30542 9/20 0.47
CALCA P06881 3/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADORA2B P29275 1/20 0.43
NAMPT P43490 1/20 0.41
EGLN1 Q9GZT9 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4068934 0.87 CALCA (0.44) ADORA2AADORA1CALCAADORA3ADORA2B
SCHEMBL4059925 0.80 CALCA (0.38) CALCAEGLN1
SCHEMBL4063494 0.68 EGLN1 (0.47) ADORA2AADORA1CALCAEGLN1L3MBTL1
SCHEMBL7687034 0.68 EGLN1 (0.66) ADORA2AADORA1EGLN1ALDH1A1
SCHEMBL14007368 0.67 EGLN1 (0.59) ADORA2AADORA1CALCAADORA3ADORA2B
SCHEMBL4061526 0.67 ADORA2A (0.53) ADORA2AADORA1CALCAADORA3ADORA2B
SCHEMBL4057517 0.67 ADORA2A (0.53) ADORA2AADORA1ADORA3ADORA2BEGLN1
SCHEMBL4062087 0.67 EGLN1 (0.58) CALCAEGLN1MAPT
SCHEMBL4060173 0.67 LMNA (0.52) CALCAEGLN1L3MBTL1LMNA
SCHEMBL4066709 0.66 EGLN1 (0.43) ADORA2AADORA1CALCAEGLN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326865-B1 AZA- AND POLYAZA-NAPHTHALENYL CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2009-05-06 EP claimed