SCHEMBL4060263

SCHEMBL4060263

Nc1ccccc1CN1CCSCC1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 1/20 0.64
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 2/20 0.51
POLB P06746 1/20 0.44
MPO P05164 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14407776 0.86 MPO (0.57) CYP2A13KDM4EALDH1A1MPOKMT2A
SCHEMBL1641681 0.82 ALDH1A1 (0.58) KDM4EALDH1A1POLBMPOMEN1
SCHEMBL2912056 0.81 ALDH1A1 (0.61) KDM4EALDH1A1POLBMPOMEN1
SCHEMBL27535071 0.79 MPO (0.46) CYP2A13KDM4EALDH1A1MPOKMT2A
SCHEMBL4764209 0.78 CYP2A13 (0.64) CYP2A13KDM4EALDH1A1
SCHEMBL4103976 0.78 CYP2A13 (1.00) CYP2A13KDM4EALDH1A1KMT2A
SCHEMBL28594898 0.78 KMT2A (0.66) CYP2A13KDM4EALDH1A1KMT2A
SCHEMBL3412153 0.78 MC4R (0.56) KDM4EALDH1A1POLBMPOKMT2A
SCHEMBL2338990 0.78 CYP2A13 (0.64) CYP2A13KDM4EALDH1A1MEN1KMT2A
SCHEMBL7510280 0.78 MPO (0.44) CYP2A13KDM4EALDH1A1POLBMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016131789-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-25 WO disclosed
EP-3056202-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-17 EP disclosed
WO-2009034390-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2009-03-19 WO disclosed