SCHEMBL4062041

SCHEMBL4062041

CC(C)c1cc(-c2ncoc2-c2ccc(CN3CCCCC3)cc2)c(OCc2ccccc2)cc1OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HRH3 Q9Y5N1 12/20 0.41
HSP90AA1 P07900 3/20 0.39
HSP90B1 P14625 1/20 0.39
TRAP1 Q12931 1/20 0.39
HSP90AB1 P08238 1/20 0.38
PDK1 Q15118 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4065754 0.99 MEN1 (0.41) MEN1KMT2AHRH3HSP90AA1HSP90B1
SCHEMBL4065747 0.93 CHKA (0.48) NPC1RAB9A
SCHEMBL4069185 0.92 HSP90AA1 (0.42) HRH3HSP90AA1HSP90B1TRAP1HSP90AB1
SCHEMBL4061207 0.92 NPC1 (0.47) MEN1KMT2AHSP90AA1NPC1RAB9A
SCHEMBL4067194 0.91 MEN1 (0.41) MEN1KMT2AHRH3NPC1RAB9A
SCHEMBL13848084 0.87 TSHR (0.46) MEN1KMT2AHRH3HSP90AA1HSP90B1
SCHEMBL4068033 0.86 MAPT (0.40)
SCHEMBL13848385 0.86 TSHR (0.44) MEN1KMT2AHRH3HSP90AA1HSP90B1
SCHEMBL4061183 0.84 NPC1 (0.41) MEN1KMT2ANPC1RAB9A
SCHEMBL4373611 0.83 FNTA (0.46) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009066060-A2 4-SUBSTITUTED-6-ISOPROPYL-BENZENE-1,3-DIOL COMPOUNDS AND THEIR USE TOPOTARGET A/S (DK) 2009-05-28 WO disclosed